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PreviewIssue DateTitleContributor(s)
JMC 2017 Volume 60 Issue 3 February (13).pdf.jpg2017Design and Synthesis of Potent and Highly Selective Orexin 1 Receptor Antagonists with a Morphinan Skeleton and Their PharmacologiesNagase, Hiroshi; Yamamoto, Naoshi; Yata, Masahiro; Ohrui, Sayaka; Okada, Takahiro; Ogawa, Yasuhiro; Hirayama, Shigeto; Kuroda, Daisuke; Watanabe, Yurie; Gouda, Hiroaki
JMC 2017 Volume 60 Issue 8 April (15).pdf.jpg2017The Identification of the Clinical Candidate (R)-(1-(4-fluorophenyl)-6-((1-methyl-1H-pyrazol-4-yl)sulfonyl)-4,4a,5,6,7,8-hexahydro-1H-pyrazolo[3,4-g]isoquinolin-4a-yl)(4-(trifluoromethyl)pyridin-2-yl)methanone (CORT125134):– A Selective Glucocorticoid RecHunt, Hazel J.; Belanoff, Joseph K.; Walters, Iain; Gourdet, Benoit; Thomas, Jennifer; Barton, Naomi; Unitt, John; Phillips, Timothy; Swift, Denise; Eaton, Emily
JMC 2017 Volume 60 Issue 8 April (13).pdf.jpg2017Enantiospecific Recognition at the A <sub>2B</sub> Adenosine Receptor by Alkyl 2-Cyanoimino-4-substituted-6-methyl-1,2,3,4-tetrahydropyrimidine-5-carboxylatesCarbajales, Carlos; Azuaje, Jhonny; Oliveira, Ana; Loza, María I.; Brea, José; Cadavid, María I.; Masaguer, Christian F.; García-Mera, Xerardo; Gutiérrez-de-Terán, Hugo; Sotelo, Eddy
JMC 2017 Volume 60 Issue 8 April (14).pdf.jpg2017Molecular basis of substrate recognition and product release by the Klebsiella pneumoniae carbapenemase (KPC-2)Pemberton, Orville Antonio; Zhang, Xiujun; Chen, Yu
JMC 2017 Volume 60 Issue 8 April (5).pdf.jpg2017Design, Synthesis, and Pharmacological Characterization of <i>N</i> -(4-(2 (6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1 <i>H</i> )yl)ethyl)phenyl)quinazolin-4-amine Derivatives: Novel Inhibitors Reversing P-Glycoprotein-Mediated Multidrug ResistanceQiu, Qianqian; Liu, Baomin; Cui, Jian; Li, Zheng; Deng, Xin; Qiang, Hao; Li, Jieming; Liao, Chen; Zhang, Bo; Shi, Wei; Pan, Miaobo; Huang, Wenlong; Qian, Hai
JMC 2017 Volume 60 Issue 8 April (4).pdf.jpg2017Emergence of Small-Molecule Non-RGD-Mimetic Inhibitors for RGD IntegrinsMiller, Lisa M.; Pritchard, John M.; Macdonald, Simon J. F.; Jamieson, Craig; Watson, Allan J. B.
JMC 2017 Volume 60 Issue 9 May (28).pdf.jpg2017Benzo-isoquinoline-diones As Potent and Selective Inhibitors of BRPF2 and TAF1/TAF1L BromodomainsBouché, Léa; Christ, Clara D.; Siegel, Stephan; Fernández-Montalván, Amaury E.; Holton, Simon J.; Fedorov, Oleg; ter Laak, Antonius; Sugawara, Tatsuo; Stöckigt, Detlef; Tallant, Cynthia; Bennett, James M.; Monteiro, Octovia P; Díaz-Sáez, Laura; Siejka, Paulina; Meier,
JMC 2017 Volume 60 Issue 9 May (3).pdf.jpg2017Diindolylmethane Derivatives – Potent Agonists of the Immunostimulatory Orphan G Protein-Coupled Receptor GPR84Pillaiyar, Thanigaimalai; Köse, Meryem; Sylvester, Katharina; Weighardt, Heike; Thimm, Dominik; Borges, Gleice; Förster, Irmgard; von Kügelgen, Ivar; Müller, Christa E
JMC 2017 Volume 60 Issue 9 May (29).pdf.jpg2017Design, Synthesis, and Biological Evaluation of Dimorpholine Substituted Thienopyrimidines as Potential Class I PI3K/mTOR Dual InhibitorsZhan, Miao; Deng, Yufang; Zhao, Lifeng; Yan, Guoyi; Wang, Fangying; Tian, Ye; Zhang, Lanxi; Jiang, Hongxia; Chen, Yuanwei
JMC 2017 Volume 60 Issue 7 April (45).pdf.jpg2017University of Michigan DRUG ANNOTATIONS EDITORS PERSPECTIVES EDITOR EDITOR EMERITUS MANAGING EDITOR EDITORIAL ADVISORY BOARDGeorg, Gunda; Wang, Shaomeng; Blagg, Brian S J; Bolognesi, Maria Laura; Conway, Stuart; Cushman, Mark; Glennon, Richard A; Garcia-echeverria, Carlos; Zablocki, Jeff; Greenlee, William J; Haskell-luevano, Carrie; Holzgrabe, Ulrike; Portoghese, Philip S; Clark, Lorraine
JMC 2017 Volume 60 Issue 5 March (41).pdf.jpg2017Members contact:-
JMC 2017 Volume 60 Issue 9 May (35).pdf.jpg2017Design of Potent and Druglike Nonphenolic Inhibitors for Catechol O-Methyltransferase Derived from a Fragment Screening Approach Targeting the S-Adenosyl- l -methionine PocketLerner, Christian; Jakob-Roetne, Roland; Buettelmann, Bernd; Ehler, Andreas; Rudolph, Markus; Sarmiento, Rosa Mar??a Rodr??guez
JMC 2017 Volume 60 Issue 4 February (30).pdf.jpg2017Members contact:-
JMC 2017 Volume 60 Issue 7 April (44).pdf.jpg2017Members contact:-
JMC 2017 Volume 60 Issue 3 February (1).pdf.jpg2017Expanding the Cancer Arsenal with Targeted Therapies: Disarmament of the Antiapoptotic Bcl ‑ 2 Proteins by Small MoleculesYap, Jeremy L; Chen, Lijia; Lanning, Maryanna E; Fletcher, Steven
JMC 2017 Volume 60 Issue 7 April (7).pdf.jpg2017Discovery of an Orally Selective Inhibitor of Signal Transducer and Activator of Transcription 3 Using Advanced Multiple Ligand Simultaneous DockingYu, Wenying; Li, Chenglong; Zhang, Wenda; Xia, Yuanzheng; Li, Shanshan; Lin, Jia Yuh; Yu, Keqin; Liu, Mu; Yang, Lei; Luo, Jianguang; Chen, Yijun; Sun, Hongbin; Kong, Lingyi
JMC 2017 Volume 60 Issue 8 April (24).pdf.jpg2017University of Michigan ASSOCIATE EDITORS DRUG ANNOTATIONS EDITORS PERSPECTIVES EDITOR EDITOR EMERITUS EDITORIAL ADVISORY BOARDGeorg, Gunda; Wang, Shaomeng; Blagg, Brian S J; Holzgrabe, Ulrike; Haskell-luevano, Carrie; Melchiorre, Carlo; Garcia-echeverria, Carlos; Zablocki, Jeff; Cushman, Mark; Glennon, Richard a; Greenlee, William J; Portoghese, Philip S; Aldrich, Courtney C; Jorgensen, Will
JMC 2017 Volume 60 Issue 9 May (22).pdf.jpg2017Prediction of antibiotic interactions using descriptors derived from compound molecular structureMason, Daniel J; Stott, Ian P; Ashenden, Stephanie Kay; Weinstein, Zohar B; Karakoc, Idil; Meral, Selin; Kuru, Nurdan; Bender, Andreas; Cokol, Murat
JMC 2017 Volume 60 Issue 9 May (23).pdf.jpg2017Transforming Sphingosine Kinase 1 Inhibitors into Dual and Sphingosine Kinase 2 Selective Inhibitors: Design, Synthesis, and in Vivo ActivityChildress, Elizabeth S.; Kharel, Yugesh; Brown, Anne M.; Bevan, David R.; Lynch, Kevin R.; Santos, Webster L.
JMC 2017 Volume 60 Issue 3 February (28).pdf.jpg2017Members contact:-