Collection home page  Journal of Medicinal Chemistry2015

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PreviewIssue DateTitleContributor(s)
2045.pdf.jpg2015Correction to Hunter−Killer Peptide (HKP) for Targeted TherapyEllerby, H. Michael; Bredesen, Dale E; Fujimura, Satoshi
2042.pdf.jpg26-Feb-2015Calbindin D28k and S100B have a similar interaction site with the lithium-inhibitable enzyme inositol monophosphatase-1: a new drug target siteAgam, Galila; Almog, Orna
2036.pdf.jpg26-Feb-2015Proteasome inhibitors with pyrazole scaffolds from structure-based virtual screeningMiller, Zachary; Kim, Keun-Sik; Lee, Do-Min; Kasam, Vinod; Baek, Si Eun; Lee, Kwang Hyun; Zhang, Yan-Yan; Ao, Lin; Carmony, Kimberly; Lee, Na-Ra; Zhou, Shou; Zhao, Qingquan; Jang, Yujin; Jeong, Hyun-Young; Zhan, Chang-Guo; Lee, Wooin; Kim, Dong-Eun; Kim, Kyung Bo
2025.pdf.jpg26-Feb-2015Prodrugs of reverse fosmidomycin analoguesBrücher, Karin; Gräwert, Tobias; Konzuch, Sarah; Held, Jana; Lienau, Claudia; Behrendt, Christoph; Illarionov, Boris; Maes, Louis; Bacher, Adelbert; Wittlin, Sergio; Mordmüller, Benjamin; Fischer, Markus; Kurz, Thomas
2015.pdf.jpg26-Feb-2015Improved synthesis of N-benzylaminoferrocene-based prodrugs and evaluation of their toxicity and antileukemic activityDaum, Steffen; Chekhun, Vasiliy F; Todor, Igor N; Lukianova, Natalia Yu; Shvets, Yulia V; Sellner, Leopold; Putzker, Kerstin; Lewis, Joe; Zenz, Thorsten; de Graaf, Inge A M; Groothuis, Geny M M; Casini, Angela; Zozulia, Oleksii; Hampel, Frank; Mokhir, Andriy
2003.pdf.jpg26-Feb-2015Folic acid-conjugated europium complexes as luminescent probes for selective targeting of cancer cellsQuici, Silvio; Casoni, Alessandro; Foschi, Francesca; Armelao, Lidia; Bottaro, Gregorio; Seraglia, Roberta; Bolzati, Cristina; Salvarese, Nicola; Carpanese, Debora; Rosato, Antonio
1992.pdf.jpg26-Feb-2015Optimization of 2-phenylcyclopropylmethylamines as selective serotonin 2C receptor agonists and their evaluation as potential antipsychotic agentsCheng, Jianjun; Giguère, Patrick M; Onajole, Oluseye K; Lv, Wei; Gaisin, Arsen; Gunosewoyo, Hendra; Schmerberg, Claire M; Pogorelov, Vladimir M; Rodriguiz, Ramona M; Vistoli, Giulio; Wetsel, William C; Roth, Bryan L; Kozikowski, Alan P
1976.pdf.jpg26-Feb-2015Discovery of highly potent, selective, and efficacious small molecule inhibitors of ERK1/2Ren, Li; Grina, Jonas; Moreno, David; Blake, James F; Gaudino, John J; Garrey, Rustam; Metcalf, Andrew T; Burkard, Michael; Martinson, Matthew; Rasor, Kevin; Chen, Huifen; Dean, Brian; Gould, Stephen E; Pacheco, Patricia; Shahidi-Latham, Sheerin; Yin, Jianping; West, Kristina; Wang, Weiru; Moffat, John G; Schwarz, Jacob B
1964.pdf.jpg26-Feb-2015Characterization of two distinct structural classes of selective aldehyde dehydrogenase 1A1 inhibitorsMorgan, Cynthia A; Hurley, Thomas D
1950.pdf.jpg26-Feb-2015Discovery and profiling of a selective and efficacious Syk inhibitorThoma, Gebhard; Smith, Alexander B; van Eis, Maurice J; Vangrevelinghe, Eric; Blanz, Joachim; Aichholz, Reiner; Littlewood-Evans, Amanda; Lee, Christian C; Liu, Hong; Zerwes, Hans-Günter
1940.pdf.jpg26-Feb-2015Antiprotozoal activity and DNA binding of dicationic acridonesMontalvo-Quirós, Sandra; Taladriz-Sender, Andrea; Kaiser, Marcel; Dardonville, Christophe
1929.pdf.jpg26-Feb-2015Structure-activity relationship of pyrrolyl diketo acid derivatives as dual inhibitors of HIV-1 integrase and reverse transcriptase ribonuclease H domainCuzzucoli Crucitti, Giuliana; Métifiot, Mathieu; Pescatori, Luca; Messore, Antonella; Madia, Valentina Noemi; Pupo, Giovanni; Saccoliti, Francesco; Scipione, Luigi; Tortorella, Silvano; Esposito, Francesca; Corona, Angela; Cadeddu, Marta; Marchand, Christophe; Pommier, Yves; Tramontano, Enzo; Costi, Roberta; Di Santo, Roberto
1915.pdf.jpg26-Feb-2015Structure-activity relationship of pyrrolyl diketo acid derivatives as dual inhibitors of HIV-1 integrase and reverse transcriptase ribonuclease H domainCuzzucoli Crucitti, Giuliana; Métifiot, Mathieu; Pescatori, Luca; Messore, Antonella; Madia, Valentina Noemi; Pupo, Giovanni; Saccoliti, Francesco; Scipione, Luigi; Tortorella, Silvano; Esposito, Francesca; Corona, Angela; Cadeddu, Marta; Marchand, Christophe; Pommier, Yves; Tramontano, Enzo; Costi, Roberta; Di Santo, Roberto
1900.pdf.jpg26-Feb-2015Novel C-4 heteroaryl 13-cis-retinamide Mnk/AR degrading agents inhibit cell proliferation and migration and induce apoptosis in human breast and prostate cancer cells and suppress growth of MDA-MB-231 human breast and CWR22Rv1 human prostate tumor xenografts in miceMbatia, Hannah W; Ramalingam, Senthilmurugan; Ramamurthy, Vidya P; Martin, Marlena S; Kwegyir-Afful, Andrew K; Njar, Vincent C O
1879.pdf.jpg26-Feb-2015Structure-activity relationship studies and in vivo activity of guanidine-based sphingosine kinase inhibitors: discovery of SphK1- and SphK2-selective inhibitorsPatwardhan, Neeraj N; Morris, Emily A; Kharel, Yugesh; Raje, Mithun R; Gao, Ming; Tomsig, Jose L; Lynch, Kevin R; Santos, Webster L
1862.pdf.jpg26-Feb-2015Discovery of 4'-chloromethyl-2'-deoxy-3',5'-di-O-isobutyryl-2'-fluorocytidine (ALS-8176), a first-in-class RSV polymerase inhibitor for treatment of human respiratory syncytial virus infectionWang, Guangyi; Deval, Jerome; Hong, Jin; Dyatkina, Natalia; Prhavc, Marija; Taylor, Joshua; Fung, Amy; Jin, Zhinan; Stevens, Sarah K; Serebryany, Vladimir; Liu, Jyanwei; Zhang, Qingling; Tam, Yuen; Chanda, Sushmita M; Smith, David B; Symons, Julian A; Blatt, Lawrence M; Beigelman, Leo
1846.pdf.jpg26-Feb-2015Bis-aryl urea derivatives as potent and selective LIM kinase (Limk) inhibitorsYin, Yan; Zheng, Ke; Eid, Nibal; Howard, Shannon; Jeong, Ji-Hak; Yi, Fei; Guo, Jia; Park, Chul Min; Bibian, Mathieu; Wu, Weilin; Hernandez, Pamela; Park, HaJeung; Wu, Yuntao; Luo, Jun-Li; LoGrasso, Philip V; Feng, Yangbo
1832.pdf.jpg26-Feb-2015Synthesis of new steroidal inhibitors of P-glycoprotein-mediated multidrug resistance and biological evaluation on K562/R7 erythroleukemia cellsde Ravel, Marc Rolland; Alameh, Ghina; Melikian, Maxime; Mahiout, Zahia; Emptoz-Bonneton, Agnès; Matera, Eva-Laure; Lomberget, Thierry; Barret, Roland; Rocheblave, Luc; Walchshofer, Nadia; Beltran, Sonia; El Jawad, Lucienne; Mappus, Elisabeth; Grenot, Catherine; Pugeat, Michel; Dumontet, Charles; Le Borgne, Marc; Cuilleron, Claude Yves
1818.pdf.jpg26-Feb-2015Structural investigation of B-Raf paradox breaker and inducer inhibitorsArora, Rohit; Di Michele, Michela; Stes, Elisabeth; Vandermarliere, Elien; Martens, Lennart; Gevaert, Kris; Van Heerde, Erika; Linders, Joannes T M; Brehmer, Dirk; Jacoby, Edgar; Bonnet, Pascal
1806.pdf.jpg26-Feb-2015Development of cyclic NGR peptides with thioether linkage: structure and dynamics determining deamidation and bioactivityEnyedi, Kata Nóra; Czajlik, András; Knapp, Krisztina; Láng, András; Majer, Zsuzsa; Lajkó, Eszter; Kőhidai, László; Perczel, András; Mező, Gábor

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